AUG 18, 2026 · JOURNAL ARTICLE
Optimizationof a Series of Novel 1 H -Pyrrolo[3,2- c ]pyridine-Based USP1Inhibitors with Potent In Vivo Antitumor Activity
Journal of Medicinal Chemistry
Early-stage preclinical chemistry and pharmacology study demonstrating lead compound design and in vivo efficacy in xenograft models, without clinical trial data or regulatory approval.
Reported
Tumor inhibition rate (38a + olap…80.7%